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Graduating School 【 display / non-display 】
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Meiji Pharmaceutical University Faculty of Pharmaceutical Science 衛生薬学科 Graduated
Graduate School 【 display / non-display 】
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Osaka University Graduate School, Division of Pharmaceutical Sciences 分子薬科学専攻 Doctor's Course Completed
Degree 【 display / non-display 】
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Meiji Pharmaceutical University -
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Osaka University - 博士（薬学）
Research field 【 display / non-display 】
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Life Science / Pharmaceutical hygiene and biochemistry (生化学、輸送体、トランスポーター)
Research Career 【 display / non-display 】
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細胞外排出型輸送体の機能と生理的役割の解明
Project Year:2003
Papers 【 display / non-display 】
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Pentafluorosulfanyl-substituted biaryl derivatives as MATE-type transporter inhibitors targeting drug-resistant bacteria
Susumu Shinya, Kentaro Kawai, Naoki Kobayashi, Yukiko Karuo, Atsushi Tarui, Kazuyuki Sato, Masato Otsuka, Masaaki Omote
Bioorganic & Medicinal Chemistry99 117606 2024.02
Joint Work
Research paper (scientific journal)
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Fluorophenylalkyl-substituted cyanoguanidine derivatives as bacteria-selective MATE transporter inhibitors for the treatment of antibiotic-resistant infections
Susumu Shinya, Kentaro Kawai, Naoki Kobayashi, Yukiko Karuo, Atsushi Tarui, Kazuyuki Sato, Masato Otsuka, Masaaki Omote
Bioorganic & Medicinal Chemistry74 117042 2022.11
Joint Work
Research paper (scientific journal)
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Importance of the Azole Moiety of Cimetidine Derivatives for the Inhibition of Human Multidrug and Toxin Extrusion Transporter 1 (hMATE1)
Susumu Shinya, Kentaro Kawai, Atsushi Tarui, Yukiko Karuo, Kazuyuki Sato, Masaya Matsuda, Kazuyuki Kitatani, Naoki Kobayashi, Takeshi Nabe, Masato Otsuka, Masaaki Omote
Chemical and Pharmaceutical Bulletin69 ( 9 ) 905 - 912 2021.09
Joint Work
Research paper (scientific journal)
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Toward the Promotion of SDGs in Kitakawachi Area -The Current Public Awareness and Possible Educational Interventions-
水野武, 小林直木, 吉田佐治子, 喜多大三, 鳥居祐介, 小野晃正, 小林俊公, 大塚正人, 藤林真美, 柳沢学
摂南大学地域総合研究所報 ( 5 ) 30 - 44 2020.03
Joint Work
Research paper (scientific journal)
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Lysophospholipid transporter and pathogenic control
Naoki Kobayashi, Yu Hisano and Tsuyoshi Nishi
Journal of Clinical and Experimental Medicine269 ( 13 ) 1082 - 1088 2019.06
Joint Work
Research paper (scientific journal)
Books 【 display / non-display 】
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A Rapid Fluorescence Assay for Measuring Sphingosine-1-Phosphate Transporter Activity in Erythrocytes (Methods in Molecular Biology)
Kobayashi, N., and Nishi, T.Scholarly book Joint author
Springer 2017.04
Review Papers 【 display / non-display 】
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サリドマイド誘導体レナリドミドの抗腫瘍効果はどのように発現するか
小林 直木
ファルマシア 50 ( 11 ) 1145 2014.11
Article, review, commentary, editorial, etc. (scientific journal) Single Work
Presentations 【 display / non-display 】
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S1P輸送体MFSD2Bのリン酸化による活性制御
日本薬学会第144年会 パシフィコ横浜 Domestic presentation Poster presentation
2024.03 -
Exploration and Synthesis of Inhibitors Targeting the Bacterial Multidrug Efflux Pump MATE-type transporter
第40回メディシナルケミストリーシンポジウム 名古屋大学（名古屋） Domestic presentation Poster presentation
2023.11 -
細菌抗菌薬排出機構MATE型輸送体の新規阻害剤の探索合成と活性評価
第46回フッ素化学討論会 枚方市総合文化芸術センター（大阪） Domestic presentation Oral presentation (general)
2023.10 -
細菌薬剤排出トランスポーターMATEを標的とした阻害剤の開発
2023年度FMODD夏の学校 大阪大学（大阪） Domestic presentation Poster presentation
2023.08 -
Development of Selective Inhibitors Targeting Multi-antimicrobial extrusion transporter to Overcome Antibiotic Resistance
23rd International Symposium on Fluorine Chemistry (ISFC) and the 9th International Symposium on Fluorous Technologies (ISoFT) Québec (Canada) International presentation Poster presentation
2023.07
Awards 【 display / non-display 】
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Ono Pharmaceutical Travel Awards
14th International Conference on Bioactive Lipids in Cancer, Inflammation, and Related Diseases Other
Country:Others
Social Activity Outside the University 【 display / non-display 】
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「夏の親子理科実験教室」における実験指導
2015.08小学生の親子を対象として、唾液からDNAを調製する実験を指導した。